[3H]Etorphine receptor binding in vivo. Small fractional occupancy elicits analgesia.
نویسندگان
چکیده
P. M. LADURON, P. F. M. JANSSEN, W. GOMMEREN, AND J. E. LEYSEN. In Vitro and in Vivo Binding Characteristics of a New Long-Acting Histamine H1 Antagonist, Astemizole 294 J. E. LEYSEN, C. J. E. NIEMEGEERS, J. M. VAN NUETEN, AND P. M. LADURON. [3H] Ketanserin (R 41 468), a Selective 3H-Ligand for Serotonin2 Receptor Binding Sites: Binding Properties, Brain Distribution, and Functional Role 301 T. A. ROBERT, A. N. HAGARDORN, AND E. A. DAIGNEAULT. Differential Stereoselectivity of Methotrimeprazine Enantiomers for Selected Central Nervous System Receptor Types 315
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عنوان ژورنال:
- Molecular pharmacology
دوره 21 2 شماره
صفحات -
تاریخ انتشار 1982